2019年度分子創薬化学セミナー(前期) - 徳島大学薬学部・大学院

第359回（2019. 9. 28）
担当者：野脇静
文献名："Asymmetric Synthesis of Alkyl Fluorides: Hydrogenation of Fluorinated Olefins"
S. Ponra, J. Yang, S. Kerdphon, and P. G. Andersson
Angew. Chem. Int. Ed., 58 (27), 9282-9287 (2019).

第358回（2019. 9. 21）
担当者：白川怜王奈
文献名："Copper-Catalyzed Radical Aminotrifluoromethylation of Alkenes"
H. Xiao, H. Shen, L. Zhu, and C. Li
J. Am. Chem. Soc., 141 (29), 11440-11445 (2019).

第357回（2019. 9. 21）
担当者：伊勢谷怜史
文献名："Direct Synthesis of Amides by Acceptorless Dehydrogenative Coupling of Benzyl Alcohols and Ammonia Catalyzed by a Manganese Pincer Complex: Unexpected Crucial Role of Base"
P. Daw, A. Kumar, N. A. Espinosa-Jalapa, Y. Ben-David, and D. Milstein
J. Am. Chem. Soc., 141 (31), 12202-12206 (2019).

第356回（2019. 7. 27）
担当者：大多和孝一
文献名："A Ten-Step Total Synthesis of Speradine C"
H. Liu, L. Chen, K. Yuan, and Y. Jia
Angew. Chem. Int. Ed., 58 (19), 6362-6365 (2019).

第355回（2019. 7. 20）
担当者：井原嵩人
文献名："Synthesis of C4-Aminated Indoles via a Catellani and Retro-Diels-Alder Strategy"
B. -S. Zhang, Y. Li, Z. Zhang, Y. An, Y. -H. Wen, X. -Y. Gou, S. -Q. Quan, X. -G. Wang, and Y. -M. Liang
J. Am. Chem. Soc., 141 (24), 9731-9738 (2019).

第354回（2019. 7. 20）
担当者：僧津真之介
文献名："A Divergent Nickel-Catalyzed Synthesis of Quinazolinediones and Benzoxazinone Imines"
W. Wertjes, S. Ayers, Q. Gao, E. M. Simmons, and G. L. Beutner
Synthesis., 50 (22), 4453-4461 (2018).

第353回（2019. 7. 6）
担当者：堀越拳
文献名："Direct Intermolecular Anti-Markovnikov Hydroazidation of Unactivated Olefins"
H. Li, S. -J. Shen, C. -L. Zhu, and H. Xu
J. Am. Chem. Soc., 141 (23), 9415-9421 (2019).

第352回（2019. 7. 6）
担当者：舟田遥乃
文献名："Dimethylprolinol Versus Diphenylprolinol in CuBr2-Catalyzed Enantioselective Allenylation of Terminal Alkynols"
D. Ma, X. Duan, C. Fu, X. Huang, and S. Ma
Synthesis., 50 (13), 2533-2545 (2018).

第351回（2019. 6. 22）
担当者：田原昌和
文献名："tert-Butoxide-Assisted Structural Transformation of 2-Aza-1,3,5-trienes: Fast Track to 5-Ethynyl-2-vinyl- and 2,5-Divinyl-1,3-thiazoles"
N. A. Nedolya, O. A. Tarasova, A. I. Albanov, and B. A. Trofimov
Synthesis., 50 (21), 4313-4324 (2018).

第350回(2019. 6. 15)
担当者:清水蘭愛
文献名:"Extending the Class of [1,3]-Dioxolo[4.5-f]benzodioxole (DBD) Fluorescent Dyes"
P. Wessig, L. John, and M. Mertens
Eur. J. Org. Chem., 2018 (14), 1674-1681 (2018).

第349回(2019. 6. 1)
担当者:仲村明人
文献名:"CuH-Catalyzed Enantioselective Alkylation of Indole Derivatives with Ligand-Controlled Regiodivergence"
Y. Ye, S. -T. Kim, J. Jeong, M. -H. Baik, and S. L. Buchwald
J. Am. Chem. Soc., 141 (9), 3901-3909 (2019).

第348回(2019. 6. 1)
担当者:岡崎遼太郎
文献名:"Regio- and Stereoselective Nickel-Catalyzed Coupling of Boronic Acids with Allenoates"
Y. Liu, M. Daka, and M. Bandini
Synthesis, 50 (16), 3187-3196 (2018).

第347回(2019. 5. 25)
担当者:戸口宗尚
文献名:"Longest C-C Single Bond among Neutral Hydrocarbons with a Bond Length beyond 1.8 Å"
Y. Ishigaki, T. Shimajiri, T. Takeda, R. Katoono, and T. Suzuki
Chem, 4 (4), 795-806 (2018).

第346回(2019. 5. 25)
担当者:今橋縁
文献名:"Dynamic Kinetic Resolution of Phosphinic Acid Derivatives via Nucleophilic Substitution at Phosphorus Center"
D. Strzelecka, O. Bak, P. Borowski, and M. Stankevic
Synthesis, 50 (24), 4922-4932 (2018).

第345回(2019. 5. 18)
担当者:原田紘之介
文献名:"N-Heterocyclic Carbene-Catalyzed Decarboxylative Alkylation of Aldehydes"
T. Ishii, Y. Kakeno, K. Nagao, and H. Ohmiya
J. Am. Chem. Soc., 141 (9), 3854-3858 (2019).

第344回(2019. 5. 18)
担当者:葉田滉大
文献名:"Trimethylphosphine-Promoted Alcoholysis of α,β-Unsaturated Imides and α,β-Unsaturated Esters"
H. Sato and S. Hosokawa
Synthesis, 50 (6), 1343-1349 (2018).

第343回(2019. 5. 11)
担当者:大多和孝一
文献名:"Ring-Opening Reactions of NHC-Boriranes with In Situ Generated HCl: Synthesis of a New Class of NHC-Boralactones"
W. Dai, S. J. Geib, and D. P. Curran
J. Am. Chem. Soc., 141 (8), 3623-3629 (2019).

第342回(2019. 5. 11)
担当者:井原嵩人
文献名:"Organocatalytic and Scalable Syntheses of Unsymmetrical 1,2,4,5-Tetrazines by Thiol-Containing Promotors"
W. Mao, W. Shi, J. Li, D. Su, X. Wang, L. Zhang, L. Pan, X. Wu, and H. Wu
Angew. Chem. Int. Ed., 58 (4), 1106-1109 (2019).

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