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2018

ペプチドへの直接的不斉反応を基盤とした非天然アミノ酸含有ペプチドの新規効率的不斉合成法開発.

猪熊 翼

Yakugaku Zasshi. 2018 , accepted.

 

A Recyclable Hydrophobic Anchor-Tagged Asymmetric Amino Thiourea Catalyst.

Takahisa Jichu, Tsubasa Inokuma, Keisuke Aihara, Taiki Kohiki, Kodai Nishida, Akira Shigenaga, Ken-ichi Yamada, and Akira Otaka,

ChemCatChem, 2018, 10 (16), 3402–3405.

 

Direct Enantioselective Indolylation of Peptidyl Imine for the Synthesis of Indolyl Glycine-Containing Peptides.

Tsubasa Inokuma, Kodai Nishida, Akira Shigenaga, Ken-ichi Yamada, and Akira Otaka,

Heterocycles, in press.

 

薬学における生命指向型化学(実用的ケミカルバイオテクノロジーの開発を目指して).

猪熊 翼、佐藤 伸一,

Yakugaku Zasshi. 2018, 138 (1), 37-38.

2017

A Convenient Method for Preparation of α-Imino Carboxylic Acid Derivatives and Application to the Asymmetric Synthesis of Unnatural α-Amino Acid Derivative.

Tsubasa Inokuma, Takahisa Jichu, Kodai Nishida, Akira Shigenaga, and Akira Otaka,

Chem. Pharm. Bull. 2017, 65 (6), 573-581.

Highlighted paper selected by Editor-in-Chief

 

Site-selective Benzoin-type Cyclization of Unsymmetrical Dialdoses Catalyzed by N-Heterocyclic Carbenes for Divergent Cyclitol Synthesis.

Bubwoong Kang, Yinli Wang, Satoru Kuwano, Yousuke Yamaoka, Kiyosei Takasu, and Ken-ichi Yamada, 

Chem. Commun. 2017, 53 (32), 4469-4472.

 

Phosphine-Promoted Migrative Cyclization of Sulfonylalkynol and Sulfonylalkynamide for the Synthesis of Oxa- and Azacycles.

Yinli Wang, Oriez Raphaël, Shogun Oh, Yasunori Miyakawa, Yousuke Yamaoka, Kiyosei Takasu, and Ken-ichi Yamada, 

Heterocycles 2017, 95 (Special Issue), 314-321.

2016

Use of a Catalytic Chiral Leaving Group for Asymmetric Substitutions at sp3-Hybridized Carbon Atoms: Kinetic Resolution of β-Amino Alcohols by p-Methoxybenzylation.

Yusuke Kuroda, Shingo Harada, Akinori Oonishi, Hiroki Kiyama, Yousuke Yamaoka, Ken-ichi Yamada, and Kiyosei Takasu, 

Angew. Chem. Int. Ed. 201655 (42), 13137-13141.

 

Desymmetrization of Acid Anhydride with Asymmetric Esterification Catalyzed by Chiral Phosphoric Acid.

Ken-ichi Yamada, Akinori Oonishi, Yusuke Kuroda, Shingo Harada, Hiroki Kiyama, Yousuke Yamaoka, and Kiyosei Takasu,

Tetrahedron Lett. 201657 (36), 4098-4100.

 

For those before 2016, see the link.